SCHEMBL6462329

SCHEMBL6462329

CCCCN(C(=O)O)C(=O)N[C@@H](CCc1ccccc1)C(=O)c1nccs1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PLA2G4A P47712 3/20 0.44
CES1 P23141 1/20 0.43
MMP2 P08253 1/20 0.43
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
CTSK P43235 1/20 0.41
F2 P00734 12/20 0.41
F10 P00742 6/20 0.41
F11 P03951 2/20 0.41
PRSS1 P07477 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464475 0.86 MMP2 (0.46) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL6467051 0.84 HPGD (0.49) MMP2MMP3MMP7CTSK
SCHEMBL7043359 0.77 MMP2 (0.42) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL6676842 0.74 CTSK (0.57) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL6467453 0.73 MMP2 (0.55) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL7048555 0.72 MMP2 (0.47) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL6464471 0.69 PLA2G4A (0.50) PLA2G4ACES1MMP2MMP3MMP7
SCHEMBL13093610 0.67 CTSS (0.55) MMP2MMP3MMP7CTSK
SCHEMBL6466424 0.67 CTSS (0.51) MMP2MMP3MMP7CTSKF2
SCHEMBL7043193 0.67 CTSS (0.51) MMP2MMP3MMP7CTSKF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed