SCHEMBL6462875

SCHEMBL6462875

O=C(O)C(c1ccccc1)C(NCc1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRB1 P18505 1/20 0.51
GABRB2 P47870 1/20 0.51
CYP2D6 P10635 2/20 0.48
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
CNR2 P34972 2/20 0.47
TDP1 Q9NUW8 1/20 0.46
AKT1 P31749 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CNR1 P21554 1/20 0.45
SLC6A9 P48067 2/20 0.44
CACNA1G O43497 1/20 0.44
ACP3 P15309 3/20 0.43
UTS2R Q9UKP6 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SLC6A5 Q9Y345 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465089 0.82 CYP2D6 (0.43) GABRB1GABRB2CYP2D6CYP1A2CYP2C19
SCHEMBL5273602 0.81 CYP1A2 (0.62) GABRB1GABRB2CYP2D6ATML3MBTL1
SCHEMBL29228705 0.79 ATM (0.52) GABRB1GABRB2CYP2D6ATML3MBTL1
SCHEMBL8430372 0.79 ACP3 (0.50) GABRB1GABRB2CYP2D6CYP1A2CYP2C19
SCHEMBL9427609 0.79 ACP3 (0.50) GABRB1GABRB2CYP2D6CYP1A2CYP2C19
SCHEMBL2487337 0.77 TDP1 (0.49) GABRB1GABRB2CYP2D6ATML3MBTL1
SCHEMBL7385115 0.77 ACP3 (0.51) GABRB1GABRB2CYP1A2CYP2C19CNR2
SCHEMBL11350168 0.76 CYP1A2 (0.56) GABRB1GABRB2CYP2D6ATML3MBTL1
SCHEMBL4237244 0.74 CYP1A2 (0.51) GABRB1GABRB2CYP2D6CYP1A2CYP2C19
SCHEMBL14099897 0.74 ACP3 (0.53) L3MBTL1TDP1ALDH1A1ACP3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
EP-1493819-A1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER Ube Industries, Ltd. (JP) 2005-01-05 EP disclosed