SCHEMBL6465089

SCHEMBL6465089

O=C(O)C(c1ccccc1)C(NCc1ccccc1)c1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.43
ACP3 P15309 4/20 0.42
GABRB1 P18505 1/20 0.41
GABRB2 P47870 1/20 0.41
VDR P11473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
ADAMTS5 Q9UNA0 1/20 0.39
HPGD P15428 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
IDO2 Q6ZQW0 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462875 0.82 GABRB1 (0.51) CYP2D6ACP3GABRB1GABRB2MEN1
SCHEMBL7785978 0.75 SMN1; SMN2 (0.49) CYP2D6VDRSMN1; SMN2MEN1KMT2A
SCHEMBL7785975 0.75 SMN1; SMN2 (0.49) CYP2D6VDRSMN1; SMN2MEN1KMT2A
SCHEMBL28525384 0.74 VDR (0.56) ACP3VDRSMN1; SMN2MEN1KMT2A
SCHEMBL7385115 0.72 ACP3 (0.51) ACP3GABRB1GABRB2SMN1; SMN2MEN1
SCHEMBL9427609 0.71 ACP3 (0.50) CYP2D6ACP3GABRB1GABRB2SMN1; SMN2
SCHEMBL8430372 0.71 ACP3 (0.50) CYP2D6ACP3GABRB1GABRB2SMN1; SMN2
SCHEMBL10763376 0.71 MMP8 (0.51) KMT2A
SCHEMBL15637982 0.69 POLB (0.52) GABRB1GABRB2SMN1; SMN2KMT2APOLB
SCHEMBL7189369 0.69 ACP3 (0.53) ACP3SMN1; SMN2MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
EP-1493819-A1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER Ube Industries, Ltd. (JP) 2005-01-05 EP disclosed