SCHEMBL6465945

SCHEMBL6465945

O=C(O)NCC(C(=O)NCCC(C(=O)c1nc2ccccc2o1)c1ccccc1)S(=O)(=O)Cc1cnccc1C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.33
GART P22102 1/20 0.33
PTPN1 P18031 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
CTSL P07711 1/20 0.32
CTSK P43235 1/20 0.32
EPHX2 P34913 1/20 0.32
PPARG P37231 1/20 0.32
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
RBP4 P02753 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CD38 P28907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7043199 0.91 SCN9A (0.35) CTSSPTPN1CTSLCTSKCYP3A4
SCHEMBL6464414 0.84 FAAH (0.38) CTSSGARTCYP3A4CYP2C9
SCHEMBL6468432 0.81 GART (0.34) CTSSGARTEPHX2CYP3A4CYP2C9
SCHEMBL6464521 0.81 CTSS (0.38) CTSSPTPN1CTSLCTSKEPHX2
SCHEMBL6465509 0.78 LMNA (0.46) CTSSCTSLEPHX2ADRB2ADRB1
SCHEMBL6062750 0.77 EPHX2 (0.38) CTSSGARTEPHX2CYP3A4CYP2C9
SCHEMBL7044860 0.77 LMNA (0.44) CTSSCTSLEPHX2ADRB2ADRB1
SCHEMBL6468407 0.76 EPHX2 (0.38) CTSSGARTEPHX2CYP3A4CYP2C9
SCHEMBL7049525 0.76 GART (0.38) CTSSGARTCYP3A4CYP2C9
SCHEMBL7043354 0.76 EPHX2 (0.39) CTSSGARTEPHX2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed