SCHEMBL6467428

SCHEMBL6467428

NC(=O)Nc1cn(-c2cc(Cl)ccc2F)nc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 1/20 0.47
KMT2A Q03164 4/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 4/20 0.38
RIPK1 Q13546 2/20 0.36
IRAK4 Q9NWZ3 2/20 0.36
NPC1 O15118 2/20 0.36
TGFBR1 P36897 1/20 0.35
TGFBR2 P37173 1/20 0.35
IKBKB O14920 1/20 0.35
SCN9A Q15858 1/20 0.35
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
KCNMA1 Q12791 1/20 0.34
GRM2 Q14416 1/20 0.34
GLA P06280 1/20 0.34
KIF11 P52732 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465833 0.80 ALDH1A1 (0.53) ITKKMT2AMEN1ALDH1A1IRAK4
SCHEMBL6468751 0.80 ITK (0.44) ITKKMT2AALDH1A1IRAK4NPC1
SCHEMBL6501912 0.79 ITK (0.52) ITKRIPK1IRAK4
SCHEMBL6504832 0.78 GRIN2B (0.41) ITKKMT2AMEN1ALDH1A1NPC1
SCHEMBL6468684 0.78 ITK (0.47) ITKKMT2AMEN1ALDH1A1IRAK4
SCHEMBL6502246 0.77 ITK (0.44) ITKALDH1A1IRAK4NPC1GAA
SCHEMBL6507842 0.76 IDO1 (0.45) ITKKMT2AMEN1ALDH1A1NPC1
SCHEMBL6498654 0.75 MAPT (0.42) ITKKMT2AMEN1ALDH1A1NPC1
SCHEMBL6499612 0.75 MARS1 (0.44) ITKKMT2AALDH1A1NPC1KDM4E
SCHEMBL6497902 0.75 SCN9A (0.43) ITKKMT2AMEN1ALDH1A1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050197338-A1 Substituted pyrazole urea compounds for the treatment of inflammation PHARMACIA AND UPJOHN COMPANY LLC 2005-09-08 US disclosed
WO-2005037797-A1 SUBSTITUTED PYRAZOLE UREA COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2005-04-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197338-A1 Substituted pyrazole urea compounds for the treatment of inflammation IL4, ARG2, CASP4 ITK 4236/4885KMT2A 3219/4885MEN1 4599/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.