SCHEMBL64675

SCHEMBL64675

CCOC(=O)C1=C(OS(=O)(=O)C(F)(F)F)CC(CO[Si](C)(C)C(C)(C)C)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
ELANE P08246 1/20 0.34
CCR5 P51681 1/20 0.34
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78189 0.91 PDK1 (0.38) PDK1PDK2PDK3PDK4CCR5
SCHEMBL78407 0.89 PDK1 (0.37) PDK1PDK2PDK3PDK4CCR5
SCHEMBL78185 0.82 PDK1 (0.40) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL65685 0.82 CHRM5 (0.40) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL65231 0.81 CHRM5 (0.39) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL18767256 0.79 RAB9A (0.43) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL8701755 0.78 PSEN1 (0.41) PDK1PDK2PDK3PDK4
SCHEMBL8701756 0.78 PSEN1 (0.41) PDK1PDK2PDK3PDK4
SCHEMBL7576828 0.77 PDK1 (0.40) PDK1PDK2PDK3PDK4ELANE
SCHEMBL4399041 0.77 TMEM97 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed