SCHEMBL78189

SCHEMBL78189

CC(=O)C1=C(OS(=O)(=O)C(F)(F)F)CC(CO[Si](C)(C)C(C)(C)C)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
PTPN1 P18031 1/20 0.34
CCR5 P51681 1/20 0.34
HTR2C P28335 1/20 0.33
PREP P48147 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL64675 0.91 PDK1 (0.38) PDK1PDK2PDK3PDK4PTPN1
SCHEMBL78407 0.89 PDK1 (0.37) PDK1PDK2PDK3PDK4PTPN1
SCHEMBL8701755 0.80 PSEN1 (0.41) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL8701756 0.80 PSEN1 (0.41) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL7576828 0.79 PDK1 (0.40) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL78185 0.76 PDK1 (0.40) PDK1PDK2PDK3PDK4
SCHEMBL78190 0.76 PDK1 (0.39) PDK1PDK2PDK3PDK4
SCHEMBL65202 0.75 MGLL (0.36) PDK1PDK2PDK3PDK4PTPN1
SCHEMBL29560191 0.75 SMN1; SMN2 (0.45) PDK1PDK2PDK3PDK4PREP
SCHEMBL78327 0.75 PDK1 (0.40) PDK1PDK2PDK3PDK4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed