SCHEMBL78185

SCHEMBL78185

CCOC(=O)C1=C(OS(=O)(=O)C(F)(F)F)CCN(C(=O)OCc2ccccc2)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
ELANE P08246 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
TSHR P16473 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL66292 0.86 ALDH1A1 (0.35) ALDH1A1MAPT
SCHEMBL64675 0.82 PDK1 (0.38) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL66854 0.81 CHRM2 (0.38) PDK1PDK2PDK3PDK4ELANE
SCHEMBL78622 0.80 SMN1; SMN2 (0.38) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL78407 0.77 PDK1 (0.37) PDK1PDK2PDK3PDK4
SCHEMBL78189 0.76 PDK1 (0.38) PDK1PDK2PDK3PDK4
SCHEMBL4399041 0.75 TMEM97 (0.45) L3MBTL1TSHR
SCHEMBL78327 0.74 PDK1 (0.40) PDK1PDK2PDK3PDK4L3MBTL1
SCHEMBL34466974 0.74 PREP (0.42) PDK1PDK2PDK3PDK4
SCHEMBL30781571 0.74 PREP (0.42) PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed