SCHEMBL65685

SCHEMBL65685

CCOC(=O)C1=C(c2ccc(O)cc2)CC(CO[Si](C)(C)C(C)(C)C)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 6/20 0.40
CHRM1 P11229 6/20 0.40
CHRM2 P08172 3/20 0.40
CHRM4 P08173 3/20 0.40
CHRM3 P20309 3/20 0.40
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
ELANE P08246 1/20 0.35
ALDH1A1 P00352 2/20 0.33
AGTR2 P50052 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65231 0.90 CHRM5 (0.39) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL78404 0.88 PDK1 (0.35) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL64233 0.86 CHRM5 (0.35) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL64056 0.86 PPARG (0.38) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL64675 0.82 PDK1 (0.38) PDK1PDK2PDK3PDK4ELANE
SCHEMBL65202 0.81 MGLL (0.36) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL66854 0.81 CHRM2 (0.38) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL8701756 0.79 PSEN1 (0.41) PDK1PDK2PDK3PDK4
SCHEMBL8701755 0.79 PSEN1 (0.41) PDK1PDK2PDK3PDK4
SCHEMBL65792 0.78 PPARA (0.39) CHRM5CHRM1ALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed