SCHEMBL6471018

SCHEMBL6471018

[c]1cc2ccccc2n1-c1cccc2ccsc12

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
DAO P14920 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28677436 0.71 BIRC5 (0.41) CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL29385772 0.71 BIRC5 (0.41) CYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL4720438 0.68 DRD2 (0.42) HTR1ADRD2
SCHEMBL718221 0.66 KDM4E (0.37)
SCHEMBL4720422 0.65 ALDH1A1 (0.45) DRD2
SCHEMBL29476084 0.65 HTR6 (0.56) SLC6A4HTR1ADRD2HTR2A
SCHEMBL13533081 0.65 HTR6 (0.56) SLC6A4HTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL30450176 0.64 LMNA (0.57) SLC6A4HTR1ADRD2HTR2A
SCHEMBL2582372 0.64 TLR9 (0.50) CYP2A6DAOHTR1ADRD2HTR2A
SCHEMBL4724581 0.63 MCHR1 (0.40) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539739-A1 PIPERIDINYL COMPOUNDS THAT SELECTIVELY BIND INTEGRINS JANSSEN PHARMACEUTICA N.V. (BE) 2005-06-15 EP disclosed
WO-2004020435-A1 PIPERIDINYL COMPOUNDS THAT SELECTIVELY BIND INTEGRINS JANSSEN PHARMACEUTICA N.V. (BE) 2004-03-11 WO disclosed