SCHEMBL6477877

SCHEMBL6477877

CC(C)(C)C[C@H](N)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
IDO1 P14902 1/20 0.47
KMT2A Q03164 2/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SLC15A1 P46059 2/20 0.45
LTA4H P09960 1/20 0.45
LAP3 P28838 1/20 0.45
SLC1A1 P43005 4/20 0.44
SLC1A3 P43003 3/20 0.44
SLC1A2 P43004 2/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28732907 1.00 ALDH1A1 (0.51) ALDH1A1CTSLCTSBCTSSIDO1
Hydrochloric Acid SCHEMBL3824193 0.98 ALDH1A1 (0.50) ALDH1A1CTSLCTSBCTSSIDO1
SCHEMBL29609090 0.85 LMNA (0.52) ALDH1A1CTSLCTSBCTSSMAPK1
SCHEMBL28962790 0.83 ALDH1A1 (0.47) ALDH1A1IDO1KMT2AMAPK1L3MBTL1
Hydrochloric Acid SCHEMBL28669155 0.83 IDO1 (0.46) ALDH1A1IDO1KMT2AMAPK1L3MBTL1
Hydrochloric Acid SCHEMBL28669153 0.83 IDO1 (0.46) ALDH1A1IDO1KMT2AMAPK1L3MBTL1
SCHEMBL23008679 0.82 ALDH1A1 (0.53) ALDH1A1CTSLCTSBCTSSKMT2A
SCHEMBL7495332 0.82 ALDH1A1 (0.53) ALDH1A1CTSLCTSBCTSSKMT2A
SCHEMBL7495338 0.82 ALDH1A1 (0.53) ALDH1A1CTSLCTSBCTSSKMT2A
SCHEMBL2130586 0.81 ALDH1A1 (0.56) ALDH1A1IDO1KMT2AMAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114681443-B Nitrile-containing antiviral compounds 辉瑞大药厂 2024-05-10 CN disclosed
CN-116789648-A Nitrile-containing antiviral compounds 辉瑞大药厂 2023-09-22 CN disclosed
CN-114466838-B Nitrile-containing antiviral compounds 辉瑞大药厂 2023-05-02 CN disclosed
EP-4166539-A1 NITRILE-CONTAINING COMPOUNDS FOR USE AS MEDICAMENTS Pfizer Inc. (US) 2023-04-19 EP disclosed
US-11541034-B2 Nitrile-containing antiviral compounds PFIZER INC. (US) 2023-01-03 US disclosed
US-11452711-B2 Nitrile-containing antiviral compounds PFIZER INC. (US) 2022-09-27 US disclosed
CN-114681443-A Nitrile-containing antiviral compounds 辉瑞大药厂 2022-07-01 CN disclosed
US-11351149-B2 Nitrile-containing antiviral compounds PFIZER INC. (US) 2022-06-07 US disclosed
US-20220142976-A1 Nitrile-Containing Antiviral Compounds PFIZER INC. (US) 2022-05-12 US disclosed
CN-114466838-A Nitrile-containing antiviral compounds 辉瑞大药厂 2022-05-10 CN disclosed
US-20050075281-A1 peptide antibiotics comprising lysobactin derivatives used for treatment and/or prophylaxis of bacterial infectious diseases; cyclic peptides BAYER HEALTHCARE AG (DE) 2005-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075281-A1 peptide antibiotics comprising lysobactin derivatives used for treatment and/or prophylaxis of bacterial infectious diseases; cyclic peptides VIP, LNPEP, HAMP ALDH1A1 4884/4885CTSL 65/4885CTSB 110/4885
US-11452711-B2 Nitrile-containing antiviral compounds ACE2, NOS2, EIF2AK2 ALDH1A1 3238/4885CTSL 635/4885CTSB 657/4885
US-20220142976-A1 Nitrile-Containing Antiviral Compounds ACE2, NOS2, EIF2AK2 ALDH1A1 3238/4885CTSL 635/4885CTSB 657/4885
US-11541034-B2 Nitrile-containing antiviral compounds ACE2, NOS2, EIF2AK2 ALDH1A1 3238/4885CTSL 635/4885CTSB 657/4885
US-11351149-B2 Nitrile-containing antiviral compounds ACE2, NOS2, EIF2AK2 ALDH1A1 3238/4885CTSL 635/4885CTSB 657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.