SCHEMBL6480023

SCHEMBL6480023

COC(=O)C1(NC(=O)C(Cl)c2ccc(OC)cc2)CCC(C)C(C)C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
CNR2 P34972 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KMT2A Q03164 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
OPRK1 P41145 1/20 0.33
EPHX2 P34913 1/20 0.33
YAP1 P46937 1/20 0.33
TEAD4 Q15561 1/20 0.33
HTT P42858 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6475667 0.91 ALDH1A1 (0.35) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL8650851 0.90 ADRA1D (0.34) ALDH1A1CYP3A4CYP2C19NPSR1PKM
SCHEMBL7961516 0.88 GPR88 (0.40) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL6474518 0.87 POLB (0.39) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL6481238 0.86 ALDH1A1 (0.36) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL6481442 0.84 SMYD3 (0.37) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL6474830 0.83 SMYD3 (0.36) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL6482178 0.82 NPSR1 (0.40) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL7675801 0.82 EPHX2 (0.37) ALDH1A1CNR2NPSR1KMT2AL3MBTL1
SCHEMBL6475209 0.82 KMT2A (0.36) ALDH1A1CYP3A4CYP2D6MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6939888-B2 1-H-3-arylpirrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 2005-09-06 US disclosed
US-20040019061-A1 1-H-3-arylpirrolidine-2,4-dione derivatives FISCHER REINER (DE) 2004-01-29 US disclosed
US-6472419-B1 1-H-3-aryl-pyrrolidine-2, 4-dione derivatives as pest-control agents BAYER AKTIENGESELLSCHAFT (DE) 2002-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040019061-A1 1-H-3-arylpirrolidine-2,4-dione derivatives PRXL2A, DDT, CYP4B1 ALDH1A1 792/4885CYP3A4 120/4885CYP2D6 416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.