SCHEMBL6483205

SCHEMBL6483205

OC[C@@H](O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.51
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
SCN9A Q15858 4/20 0.43
PNMT P11086 1/20 0.42
ACP3 P15309 1/20 0.42
PDE2A O00408 2/20 0.41
ORAI1 Q96D31 1/20 0.40
ORAI2 Q96SN7 1/20 0.40
ORAI3 Q9BRQ5 1/20 0.40
TRPV6 Q9H1D0 1/20 0.40
KIF11 P52732 1/20 0.40
MGLL Q99685 1/20 0.40
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17663780 1.00 HSD11B1 (0.51) HSD11B1CES2CES1SCN9APNMT
SCHEMBL1155302 1.00 HSD11B1 (0.51) HSD11B1CES2CES1SCN9APNMT
SCHEMBL13285842 0.83 HSD11B1 (0.49) HSD11B1CES2CES1PNMTACP3
SCHEMBL17987913 0.83 HSD11B1 (0.51) HSD11B1CES2CES1PNMTACP3
SCHEMBL25159746 0.81 HSD11B1 (0.50) HSD11B1CES2CES1PNMTACP3
SCHEMBL7153429 0.81 PNMT (0.62) HSD11B1CES2CES1PNMTACP3
SCHEMBL18285644 0.81 HSD11B1 (0.50) HSD11B1CES2CES1PNMTACP3
SCHEMBL4292372 0.81 PNMT (0.62) HSD11B1CES2CES1PNMTACP3
SCHEMBL7783843 0.81 HSD11B1 (0.50) HSD11B1CES2CES1PNMTACP3
SCHEMBL478137 0.81 PDE2A (0.56) HSD11B1CES2CES1PNMTACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160097063-A1 Production Of Enantiopure alpha-Hydroxy Carboxylic Acids From Alkenes By Cascade Biocatalysis NATIONAL UNIVERSITY OF SINGAPORE (SG) 2016-04-07 US disclosed
US-20050004161-A1 4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxamides as antiviral agents AGOURON PHARMACEUTICALS, INC. 2005-01-06 US disclosed
US-20040249220-A1 Process for producing optically active 2-alkoxy-1-(trifluoromethyl-substituted phenyl) ethanol derivatives CENTRAL GLASS COMPANY, LIMITED (JP) 2004-12-09 US disclosed
WO-2004037760-A2 PROCESS FOR PRODUCING OPTICALLY ACTIVE 2-ALKOXY-1-(TRIFLUOROMETHYL-SUBSTITUTED PHENYL)ETHANOL DERIVATIVES CENTRAL GLASS COMPANY, LIMITED (JP) 2004-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004161-A1 4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carboxamides as antiviral agents ZC3HAV1, IRF3, BRD4 HSD11B1 3772/4885CES2 1710/4885CES1 1726/4885
US-20040249220-A1 Process for producing optically active 2-alkoxy-1-(trifluoromethyl-substituted phenyl) ethanol derivatives ADH1A, ADH1C, ADH5 HSD11B1 108/4885CES2 115/4885CES1 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.