SCHEMBL648905

SCHEMBL648905

CCCCn1c(-c2ccccc2C)nc(-c2ccccc2)c1CC(CC(C)C)NCc1ccc(C(=O)OC)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
KMT2A Q03164 1/20 0.35
AGTR1 P30556 5/20 0.34
MME P08473 4/20 0.34
F2 P00734 1/20 0.34
F7 P08709 1/20 0.34
F3 P13726 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
TLR7 Q9NYK1 1/20 0.34
ACAT1 P24752 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652578 0.95 AGTR1 (0.34) RARARARBRARGAGTR1MME
SCHEMBL650059 0.89 AGTR1 (0.37) AGTR1MME
SCHEMBL652331 0.88 DRD2 (0.35) AGTR1
SCHEMBL648189 0.88 DRD2 (0.34) AGTR1
SCHEMBL652770 0.87 TLR8 (0.35) AGTR1F2F7F3
SCHEMBL650291 0.86 DRD2 (0.33) MEN1KMT2AAGTR1
SCHEMBL651121 0.82 MEN1 (0.34) MEN1KMT2AAGTR1
SCHEMBL648999 0.82 ADORA3 (0.37) RARARARBRARGMEN1KMT2A
SCHEMBL648906 0.80 HDAC1 (0.39) KMT2AAGTR1TLR7HDAC1
SCHEMBL650281 0.80 AGTR1 (0.40) AGTR1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed