SCHEMBL650059

SCHEMBL650059

CCCCn1c(-c2ccccc2C)nc(-c2ccc(C)cc2)c1CC(CC(C)C)NCc1ccc(C(=O)O)cc1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 15/20 0.37
MME P08473 13/20 0.37
ADORA3 P0DMS8 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
AGTR2 P50052 1/20 0.35
NR1H4 Q96RI1 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL648999 0.93 ADORA3 (0.37) AGTR1ADORA3ADORA2BADORA1AGTR2
SCHEMBL652578 0.92 AGTR1 (0.34) AGTR1MME
SCHEMBL650087 0.90 ADORA3 (0.35) AGTR1ADORA3ADORA2BADORA1AGTR2
SCHEMBL648905 0.89 RARA (0.35) AGTR1MME
SCHEMBL651281 0.89 ADORA3 (0.37) AGTR1MMEADORA3ADORA2BADORA1
SCHEMBL650385 0.87 ADORA3 (0.36) AGTR1ADORA3ADORA2BADORA1AGTR2
SCHEMBL652331 0.85 DRD2 (0.35) AGTR1ADORA2B
SCHEMBL648189 0.85 DRD2 (0.34) AGTR1ADORA2B
SCHEMBL652770 0.84 TLR8 (0.35) AGTR1
SCHEMBL651079 0.84 AGTR1 (0.34) AGTR1MMEADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed