SCHEMBL6492415

SCHEMBL6492415

CC1CC(c2c[nH]c3c(F)c(F)ccc23)=CCN1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.42
HTR2A P28223 1/20 0.41
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6497949 0.77 TDO2 (0.46)
SCHEMBL6491562 0.76 AR (0.40) ARHTR2AHTR1D
SCHEMBL6812096 0.74 HTR2C (0.55) ARHTR2AHTR1D
SCHEMBL4788776 0.71 IDH1 (0.36)
SCHEMBL6492320 0.69 HTR1D (0.37) ARHTR2AHTR1D
SCHEMBL31358140 0.69 HTR2A (0.53) ARHTR2A
SCHEMBL7205820 0.69 SLC6A4 (0.53) HTR2AHTR1D
SCHEMBL6625901 0.69 HTR2C (0.41) HTR2AHTR1D
Hydrochloric Acid SCHEMBL6335001 0.67 HTR2C (0.31)
SCHEMBL1078755 0.66 HTR7 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6844338-B2 Piperidyindoles as serotonin receptor ligands ELI LILLY AND COMPANY (US) 2005-01-18 US disclosed
US-20030225068-A1 Piperidyindoles as serotonin receptor ligands ELI LILLY AND COMPANY 2003-12-04 US disclosed
EP-1286992-A1 PIPERIDYINDOLES AS SEROTONIN RECEPTOR LIGANDS ELI LILLY AND COMPANY (US) 2003-03-05 EP disclosed
WO-2001087881-A1 PIPERIDYINDOLES AS SEROTONIN RECEPTOR LIGANDS ELI LILLY AND COMPANY (US) 2001-11-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225068-A1 Piperidyindoles as serotonin receptor ligands CNR1, HTR1D, HTR1A AR 299/4885HTR2A 24/4885HTR1D 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.