SCHEMBL6494288

SCHEMBL6494288

O=C(O)[C@H](Cc1ccc2oc(CCCNc3ccccn3)cc(=O)c2c1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.52
ITGAV P06756 12/20 0.52
ITGA2B P08514 9/20 0.52
ITGB1 P05556 6/20 0.50
ITGA5 P08648 6/20 0.50
MDM4 O15151 1/20 0.41
MDM2 Q00987 1/20 0.41
MMP2 P08253 2/20 0.41
ADAMTS4 O75173 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
MMP9 P14780 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204669 0.91 ITGB1 (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL3041592 0.89 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6496052 0.88 ITGB1 (0.47) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL5204428 0.88 ITGB1 (0.47) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL13170303 0.87 ITGB1 (0.51) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6505728 0.87 ITGB3 (0.49) ITGB3ITGAVITGA2BMMP2ADAMTS4
SCHEMBL13170301 0.85 ITGB1 (0.53) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL13170302 0.83 ITGB1 (0.49) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL6503005 0.82 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB1ITGA5
SCHEMBL3048694 0.82 ITGB1 (0.50) ITGB3ITGAVITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed