Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL6494737

COc1ccc(-c2nc(C(=O)NCc3cc(CC(OC(C)C)C(=O)O)ccn3)c(C)s2)cc1.O=C(O)C(F)(F)F

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 19/20 0.44
PPARD Q03181 13/20 0.41
PPARG P37231 15/20 0.41
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6505042 0.93 PPARA (0.42) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6531504 0.92 PPARA (0.40) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6504387 0.91 PPARA (0.42) PPARAPPARDPPARG
SCHEMBL6494741 0.89 PPARA (0.39) PPARAPPARDPPARGGSK3B
Trifluoroacetic Acid SCHEMBL6498705 0.88 PPARA (0.37) PPARAPPARDPPARGGSK3B
Trifluoroacetic Acid SCHEMBL6499170 0.87 ADORA2A (0.39) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6503592 0.85 KDM4E (0.37) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6505587 0.84 PPARA (0.38) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6495816 0.84 SHMT1 (0.44) PPARAPPARDPPARG
SCHEMBL6531507 0.82 PARP1 (0.36) PPARAPPARDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed