Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL6499170

COc1ccccc1-c1nc(C(=O)NCc2cc(CC(OC(C)C)C(=O)O)ccn2)c(C)s1.O=C(O)C(F)(F)F

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.39
ADORA1 P30542 2/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
KDM4E B2RXH2 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
PPARA Q07869 7/20 0.37
PPARD Q03181 5/20 0.37
PPARG P37231 4/20 0.37
MAPT P10636 3/20 0.37
SHMT2 P34897 2/20 0.37
KDM1A O60341 1/20 0.36
HDAC1 Q13547 1/20 0.36
LMNA P02545 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6505587 0.90 PPARA (0.38) ADORA2AADORA1ALDH1A1HPGDPPARA
Trifluoroacetic Acid SCHEMBL6531504 0.90 PPARA (0.40) PPARAPPARDPPARGMAPT
SCHEMBL6499174 0.90 ADORA1 (0.38) ADORA2AADORA1ALDH1A1HPGDHSD17B10
Trifluoroacetic Acid SCHEMBL6494737 0.87 PPARA (0.44) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6505042 0.86 PPARA (0.42) ALDH1A1HPGDKDM4EPPARAPPARD
Trifluoroacetic Acid SCHEMBL6495816 0.85 SHMT1 (0.44) KDM4EPPARAPPARDPPARGMAPT
Trifluoroacetic Acid SCHEMBL6503592 0.85 KDM4E (0.37) ALDH1A1KDM4EPPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6504387 0.84 PPARA (0.42) PPARAPPARDPPARG
Trifluoroacetic Acid SCHEMBL6498705 0.81 PPARA (0.37) PPARAPPARDPPARG
SCHEMBL6531507 0.80 PARP1 (0.36) ADORA2AALDH1A1HPGDKDM4EPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed