SCHEMBL6494741

SCHEMBL6494741

COc1ccc(-c2nc(C(=O)NCc3cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn3)c(C)s2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.39
GSK3B P49841 2/20 0.37
PPARD Q03181 3/20 0.36
CDK2 P24941 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
PPARG P37231 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
WDR5 P61964 4/20 0.35
MAPT P10636 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505045 0.93 SMN1; SMN2 (0.35) PPARAPPARDADORA2AADORA1PPARG
SCHEMBL6504395 0.92 PPARA (0.37) PPARAGSK3BPPARDCDK2PPARG
SCHEMBL6531507 0.91 PARP1 (0.36) PPARAPPARDADORA2APPARGADORA3
Trifluoroacetic Acid SCHEMBL6494737 0.89 PPARA (0.44) PPARAGSK3BPPARDPPARG
SCHEMBL6498709 0.88 CDK2 (0.34) PPARAGSK3BPPARDCDK2WDR5
SCHEMBL6499174 0.87 ADORA1 (0.38) ADORA2AADORA1ADORA3KMT2AGAA
SCHEMBL6503597 0.85 KDM4E (0.36) KMT2AGAAMAPTHDAC3HDAC1
SCHEMBL6505593 0.85 ADORA2A (0.35) PPARAPPARDADORA2AADORA1ADORA3
SCHEMBL6495822 0.84 SHMT1 (0.39) KMT2AWDR5MAPT
Trifluoroacetic Acid SCHEMBL6505042 0.82 PPARA (0.42) PPARAPPARDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed