SCHEMBL6497810

SCHEMBL6497810

C1=CN(C2CCNCC2)CN1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28045452 0.80
SCHEMBL27257119 0.75 GAA (0.33) ALOX15
SCHEMBL28120282 0.74 MEN1 (0.32) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL10767394 0.68
SCHEMBL4890557 0.67 HTR6 (0.34)
SCHEMBL27729342 0.67 HTR2C (0.33) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL27895099 0.65 HTR2C (0.33) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL6489205 0.65
SCHEMBL28281585 0.64 MEN1 (0.31) MEN1ALDH1A1MAPTPKMALOX15
SCHEMBL27266578 0.64 MEN1 (0.34) MEN1ALDH1A1MAPTPKMALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1026588-C 1-alkyl substituted benzimidazole derivatives, process for preparing same and pharmaceutical composition containing same JANSSEN PHARMACEUTICA NV (BE) 1994-11-16 CN claimed
CN-88101286-A 1-alkyl substituted benzimidazole derivatives, process for preparing same and pharmaceutical composition containing same 1988-09-28 CN claimed
CN-116947852-A Synthesis method of zimetapam intermediate 南通常佑药业科技有限公司 2023-10-27 CN disclosed
CN-107428744-A Novel heterocyclic compounds and its application in medicine and cosmetics 盖尔德马研究及发展公司 2017-12-01 CN disclosed
CN-106432232-A Synthesis method of 1-piperidin-4-yl-1,3-dihydro-imidazol[4, 5-b]pyridine-2-one 苏州汉德创宏生化科技有限公司 2017-02-22 CN disclosed
CN-106061969-A TRPA1 modulators 阿尔戈么迪克斯有限公司 2016-10-26 CN disclosed
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2005-11-17 US disclosed
EP-1163239-A1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055154-A1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed
CN-1026588-C 1-alkyl substituted benzimidazole derivatives, process for preparing same and pharmaceutical composition containing same JANSSEN PHARMACEUTICA NV (BE) 1994-11-16 CN disclosed
CN-1018614-B Process for preparing antihistaminic compositions containing N-heterocyclyl-4-piperidinamines JANSSEN PHARMACEUTICA NV (BE) 1992-10-14 CN disclosed
CN-88101286-A 1-alkyl substituted benzimidazole derivatives, process for preparing same and pharmaceutical composition containing same 1988-09-28 CN disclosed
CN-87100563-A The anti-histamine compositions that contains N-heterocyclic radical-4-piperidinamines 1987-08-19 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity GPR119, GIPR, PGC MEN1 1397/4885ALDH1A1 2202/4885MAPT 3231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.