SCHEMBL6499174

SCHEMBL6499174

COc1ccccc1-c1nc(C(=O)NCc2cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn2)c(C)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.38
ADORA2A P29274 2/20 0.38
ALDH1A1 P00352 7/20 0.36
MAPT P10636 5/20 0.36
NPSR1 Q6W5P4 3/20 0.36
KDM4E B2RXH2 7/20 0.36
HSD17B10 Q99714 6/20 0.36
HPGD P15428 6/20 0.36
KDM1A O60341 1/20 0.35
HDAC1 Q13547 1/20 0.35
LMNA P02545 1/20 0.34
WDR5 P61964 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
THRB P10828 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505593 0.90 ADORA2A (0.35) ADORA1ADORA2AALDH1A1KDM4EHPGD
Trifluoroacetic Acid SCHEMBL6499170 0.90 ADORA2A (0.39) ADORA1ADORA2AALDH1A1MAPTNPSR1
SCHEMBL6531507 0.89 PARP1 (0.36) ADORA2AALDH1A1MAPTKDM4EHPGD
SCHEMBL6494741 0.87 PPARA (0.39) ADORA1ADORA2AMAPTHDAC1WDR5
SCHEMBL6505045 0.86 SMN1; SMN2 (0.35) ADORA1ADORA2AALDH1A1KDM4EHPGD
SCHEMBL6495822 0.85 SHMT1 (0.39) MAPTKDM4EHPGDWDR5KMT2A
SCHEMBL6503597 0.85 KDM4E (0.36) ALDH1A1MAPTNPSR1KDM4EHDAC1
SCHEMBL6504395 0.85 PPARA (0.37) MAPTWDR5SMN1; SMN2GAA
SCHEMBL6498709 0.82 CDK2 (0.34) MAPTWDR5NPC1
Trifluoroacetic Acid SCHEMBL6505587 0.80 PPARA (0.38) ADORA1ADORA2AALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed