SCHEMBL6504471

SCHEMBL6504471

O=[N+]([O-])c1ccc(CCc2ccccc2S(=O)(=O)c2ccccc2CCc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KCNJ1 P48048 2/20 0.44
KCNH2 Q12809 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.43
HTT P42858 1/20 0.43
PTPRF P10586 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN11 Q06124 1/20 0.43
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
CA12 O43570 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
CA4 P22748 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
BCHE P06276 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11104408 0.80 ALDH1A1 (0.55) TSHRMEN1KMT2AKCNJ1KCNH2
SCHEMBL6504475 0.78 TSHR (0.60) TSHRKMT2AKCNJ1KCNH2LOXL2
SCHEMBL13946243 0.77 CYP1A2 (0.67) TSHRMEN1KMT2AKCNJ1KCNH2
SCHEMBL3292782 0.77 TSHR (0.75) TSHRKCNJ1KCNH2CYP1A2CYP2C19
SCHEMBL27583120 0.75 ALDH1A1 (0.65) TSHRMEN1KMT2AKCNJ1KCNH2
SCHEMBL3672572 0.75 HSD11B1 (0.55) MEN1KMT2ACA1CA2ALDH1A1
SCHEMBL28299042 0.74 CA12 (0.47) TSHRMEN1KMT2ACYP1A2CYP2C19
SCHEMBL4661774 0.74 CA2 (0.57) MEN1KMT2ACYP1A2CYP2C19LOXL2
SCHEMBL4618998 0.74 MMP2 (0.49) MEN1KMT2AALDH1A1
SCHEMBL11842004 0.72 KMT2A (0.61) MEN1KMT2AHTTCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005103035-A1 MODIFIED FISCHER INDOLE SYNTHESIS OF ELETRIPTAN PFIZER LIMITED (GB) 2005-11-03 WO disclosed