SCHEMBL6505102

SCHEMBL6505102

NC(=O)N(OC(=O)C(F)(F)F)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.37
NPSR1 Q6W5P4 1/20 0.35
MLYCD O95822 2/20 0.35
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ATM Q13315 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
POLB P06746 1/20 0.32
PARP1 P09874 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28173074 0.87 ALDH1A1 (0.43) CES1NPSR1MLYCDALDH1A1TDP1
SCHEMBL27659173 0.83 KMT2A (0.34) CES1ALDH1A1TDP1L3MBTL1MEN1
SCHEMBL28760313 0.83 KIF11 (0.41) CES1ALDH1A1TDP1KMT2A
SCHEMBL6506843 0.83 KCNN4 (0.41) CES1KMT2APARP1KCNN4
Water SCHEMBL10825040 0.82 CES1 (0.34) CES1NPSR1MLYCDALDH1A1TDP1
SCHEMBL27659169 0.82 HTR3E (0.41) NPSR1ALDH1A1POLBPARP1MAPT
SCHEMBL27659171 0.82 CES2 (0.41) NPSR1ALDH1A1MAPTTSHR
SCHEMBL27659195 0.80 PARP15 (0.39) MLYCDNR1H3
SCHEMBL11141452 0.80 NPSR1 (0.41) NPSR1ALDH1A1TDP1L3MBTL1ATM
SCHEMBL6012131 0.79 NPSR1 (0.38) CES1NPSR1MLYCDALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO claimed
CN-1859912-A Inhibitors of Akt activity SMITHKLINE BEECHAM CORP (US) 2006-11-08 CN disclosed