SCHEMBL6506843

SCHEMBL6506843

NC(=O)N(OC(=O)C(F)(F)F)c1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.41
PARP1 P09874 1/20 0.40
USP2 O75604 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGIR P43119 5/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
PKM P14618 1/20 0.35
CETP P11597 2/20 0.34
PTGDR Q13258 2/20 0.34
PTGER4 P35408 1/20 0.34
PTGER3 P43115 1/20 0.34
PTGER2 P43116 1/20 0.34
MAOB P27338 1/20 0.33
PARP10 Q53GL7 1/20 0.33
LIPE Q05469 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27659169 0.84 HTR3E (0.41) PARP1PTGIRCETPPTGDRLIPE
SCHEMBL27659171 0.84 CES2 (0.41) CES2PKMMAOB
SCHEMBL6505102 0.83 CES1 (0.37) KCNN4PARP1KMT2ACES1
SCHEMBL27659153 0.81 PDK1 (0.37) KCNN4KMT2A
SCHEMBL28757754 0.74 RXRA (0.38)
SCHEMBL27659173 0.74 KMT2A (0.34) KMT2ACES2CES1
SCHEMBL28760313 0.74 KIF11 (0.41) KMT2ACES2CES1MAOB
SCHEMBL28173074 0.71 ALDH1A1 (0.43) KMT2ACES1
SCHEMBL6486260 0.71 PARP1 (0.50) KCNN4PARP1KMT2ACES2CES1
SCHEMBL27659195 0.71 PARP15 (0.39) PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO claimed