SCHEMBL6505176

SCHEMBL6505176

COC(=O)CC(C)C(=NOCc1ccc(C)cc1)c1ccc(O)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.43
RAB9A P51151 5/20 0.40
NPC1 O15118 4/20 0.40
MAPT P10636 4/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPK1 P28482 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
ESRRB O95718 1/20 0.37
MAOB P27338 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
KMT2A Q03164 2/20 0.36
PARP10 Q53GL7 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507732 0.89 RAB9A (0.47) RAB9ANPC1MAPTALDH1A1MAPK1
SCHEMBL6507906 0.89 S1PR1 (0.43) S1PR1MAPTALDH1A1MAPK1PPARG
SCHEMBL6507739 0.81 GRM5 (0.42) RAB9ANPC1MAPTPPARGPPARA
SCHEMBL6533650 0.77 MAOB (0.42) S1PR1RAB9ANPC1MAPTESRRB
SCHEMBL6510873 0.77 PPARG (0.46) S1PR1RAB9ANPC1PPARGPPARA
SCHEMBL9734549 0.72 CA1 (0.48) ALDH1A1ESRRBL3MBTL1TDP1KMT2A
SCHEMBL6505172 0.68 ESR1 (0.47) S1PR1PPARGPPARAL3MBTL1KMT2A
SCHEMBL13057604 0.67 ALDH1A1 (0.57) RAB9ANPC1MAPTALDH1A1MAPK1
SCHEMBL12637601 0.67 NPC1 (0.71) RAB9ANPC1MAPTALDH1A1L3MBTL1
SCHEMBL12137308 0.67 NPC1 (0.71) RAB9ANPC1MAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040127-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2005-05-06 WO disclosed