SCHEMBL6506624

SCHEMBL6506624

O=C(Nc1nc2ccccc2[nH]1)c1ccc(CNc2ccc(-c3nc4ccccc4[nH]3)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 3/20 0.68
MMP2 P08253 2/20 0.64
MMP9 P14780 2/20 0.64
MMP8 P22894 2/20 0.64
MMP13 P45452 2/20 0.64
NPC1 O15118 8/20 0.62
RAB9A P51151 8/20 0.62
PKM P14618 4/20 0.62
KLF5 Q13887 2/20 0.62
HDAC1 Q13547 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.58
MAOB P27338 1/20 0.58
ADORA2A P29274 1/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
KDM4E B2RXH2 3/20 0.57
SCD O00767 1/20 0.57
OPRK1 P41145 1/20 0.57
TP53 P04637 1/20 0.57
HSD17B10 Q99714 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6514739 0.89 MMP2 (0.80) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6511104 0.88 HPSE (0.72) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6506903 0.88 HPSE (0.72) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6530461 0.86 KDM4E (0.70) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6527951 0.85 HPSE (0.61) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6529482 0.84 HPSE (0.59) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6532397 0.84 NPC1 (0.65) HPSENPC1RAB9AHDAC1SMN1; SMN2
SCHEMBL6281518 0.82 HPSE (1.00) HPSEMMP2MMP9MMP8MMP13
SCHEMBL8820125 0.82 HPSE (1.00) HPSEMMP2MMP9MMP8MMP13
SCHEMBL11703736 0.79 NPC1 (0.91) NPC1RAB9APKMKLF5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042496-A1 (BENZIMIDAZOL-2-YL)-PHENYL-BENZYL-AMINE DERIVATIVES AND METHODS FOR INHIBITING HEPARANASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-05-12 WO disclosed