SCHEMBL6527951

SCHEMBL6527951

NC(=O)c1ccc(CNc2ccc(-c3nc4ccccc4[nH]3)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 3/20 0.61
HDAC3 O15379 1/20 0.57
PARP1 P09874 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC2 Q92769 1/20 0.57
PARP2 Q9UGN5 1/20 0.57
MMP2 P08253 3/20 0.56
MMP9 P14780 3/20 0.56
MMP8 P22894 3/20 0.56
MMP13 P45452 3/20 0.56
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
HPGD P15428 2/20 0.55
KMT2A Q03164 1/20 0.55
NPC1 O15118 1/20 0.55
LMNA P02545 1/20 0.55
PKM P14618 1/20 0.55
NFKB1 P19838 1/20 0.55
RAB9A P51151 1/20 0.55
NFKB2 Q00653 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530461 0.90 KDM4E (0.70) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6529482 0.88 HPSE (0.59) HPSEMMP2MMP9MMP8MMP13
SCHEMBL3663760 0.85 KDM4E (0.73) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6506624 0.85 HPSE (0.68) HPSEHDAC3PARP1HDAC1HDAC2
SCHEMBL6527955 0.84 NPC1 (0.69) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6514739 0.84 MMP2 (0.80) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6529214 0.84 HPSE (0.60) HPSEKDM4EALDH1A1KMT2ANPC1
SCHEMBL6511104 0.83 HPSE (0.72) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6506903 0.83 HPSE (0.72) HPSEMMP2MMP9MMP8MMP13
SCHEMBL6533101 0.82 NPC1 (0.56) HPSEMMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042496-A1 (BENZIMIDAZOL-2-YL)-PHENYL-BENZYL-AMINE DERIVATIVES AND METHODS FOR INHIBITING HEPARANASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-05-12 WO disclosed