SCHEMBL6506915

SCHEMBL6506915

O=CC(c1ccc(F)cc1)N1CC(F)(CS(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
USP2 O75604 1/20 0.33
CRBN Q96SW2 1/20 0.32
TP53 P04637 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
MMP2 P08253 2/20 0.31
MMP9 P14780 1/20 0.31
MMP14 P50281 1/20 0.31
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5189110 0.99 LMNA (0.32) LMNAUSP2CRBNTP53HTR2A
SCHEMBL1122123 0.78 CYP3A4 (0.43) USP2MAPTPKM
SCHEMBL5189063 0.76 MMP2 (0.40) LMNAUSP2CRBNTP53HTR2A
SCHEMBL5827168 0.68 ALDH1A1 (0.48) USP2HTR2AHTR2CCA1CA2
Hydrochloric Acid SCHEMBL1121811 0.67 ALDH1A1 (0.47) USP2HTR2AHTR2CMAPTPKM
SCHEMBL17101994 0.66 PKM (0.48) USP2PKM
Hydrochloric Acid SCHEMBL5787327 0.65 AOC2 (0.34) HTR2AHTR2CMAPT
SCHEMBL3244612 0.64 SLC6A2 (0.45)
Hydrochloric Acid SCHEMBL3997950 0.63 SLC6A2 (0.44)
Hydrochloric Acid SCHEMBL3252467 0.63 SLC6A2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005047247-A1 NOVEL1,3-DISUBSTITUTED AZETIDINE DERIVATIVES FOR USE AS 5HT2A RECEPTOR LIGANDS MERCK SHARP & DOHME LIMITED (GB) 2005-05-26 WO claimed