SCHEMBL6508602

SCHEMBL6508602

O=C(O)[C@@H]1CCCN1Cc1ccc(OCc2cccc(Cl)c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.65
MAOA P21397 4/20 0.65
S1PR1 P21453 1/20 0.63
S1PR5 Q9H228 1/20 0.63
SPHK1 Q9NYA1 5/20 0.62
SPHK2 Q9NRA0 4/20 0.61
CD274 Q9NZQ7 4/20 0.60
PDCD1 Q15116 2/20 0.60
RXRA P19793 1/20 0.55
RXRB P28702 1/20 0.55
RXRG P48443 1/20 0.55
SCN3A Q9NY46 1/20 0.53
POLB P06746 1/20 0.52
GID4 Q8IVV7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6508605 1.00 MAOB (0.65) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL6167500 0.90 MAOB (0.79) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL6167507 0.90 MAOB (0.79) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL6171507 0.88 MAOA (0.61) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL3148367 0.87 NPBWR1 (0.53) SPHK1CD274PDCD1
SCHEMBL1815987 0.87 NPBWR1 (0.53) SPHK1CD274PDCD1
SCHEMBL2030130 0.87 NPBWR1 (0.53) SPHK1CD274PDCD1
SCHEMBL6171239 0.87 MAOB (0.74) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL6171245 0.87 MAOB (0.74) MAOBMAOAS1PR1S1PR5SPHK1
SCHEMBL7814221 0.84 NPBWR1 (0.58) CD274PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040108-A1 PROLINAMIDE DERIVATIVES AS SODIUM AND/OR CALCIUM CHANNEL BLOCKERS OR SELECTIVE MAO-B INHIBITORS NEWRON PHARMACEUTICALS S.P.A. (IT) 2005-05-06 WO claimed
WO-2005037828-A1 NOVEL INHIBITORS OF DPP-IV, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD. (KR) 2005-04-28 WO disclosed