SCHEMBL6509590

SCHEMBL6509590

O=C(Nc1nc2c(CCN3CCOCC3)cccc2[nH]c1=O)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 3/20 0.47
HTR1A P08908 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
KCNH2 Q12809 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
EPHX2 P34913 2/20 0.44
GAA P10253 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PARP1 P09874 3/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
HTR3A P46098 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504605 0.91 USP2 (0.44) KDM4EALDH1A1NPC1RAB9AEPHX2
SCHEMBL6505871 0.91 PARP1 (0.45) KDM4ENPSR1ALDH1A1GAAHSD17B10
SCHEMBL6508473 0.87 MAPK1 (0.46) KDM4EALDH1A1RAB9AGAAHSD17B10
SCHEMBL17731555 0.71 IRAK4 (0.56) KDM4EALDH1A1NPC1RAB9AGAA
SCHEMBL6532182 0.71 KDM4E (0.77) KDM4ENPSR1ALDH1A1HTR1AMAOA
SCHEMBL6644132 0.71 RAB9A (0.43) KDM4EALDH1A1RAB9AGAAHSD17B10
Hydrochloric Acid SCHEMBL8814898 0.67 GRIN2B (0.59) KDM4EALDH1A1HTR1ANPC1RAB9A
SCHEMBL6530642 0.66 KDM4E (1.00) KDM4ENPSR1ALDH1A1RAB9AHSD17B10
Moclobemide SCHEMBL3408310 0.66 CD274 (1.00) KDM4EALDH1A1HTR1AMAOAMAOB
Moclobemide SCHEMBL49708 0.66 CD274 (1.00) KDM4EALDH1A1HTR1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed