SCHEMBL6509836

SCHEMBL6509836

CN(C(=O)c1cc(C(N)=O)c(NC(N)=O)s1)c1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.48
HSD17B2 P37059 2/20 0.48
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
TDP1 Q9NUW8 2/20 0.47
MAPT P10636 1/20 0.47
IKBKB O14920 11/20 0.46
JAK2 O60674 2/20 0.46
JAK3 P52333 1/20 0.46
CHEK1 O14757 4/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.42
EIF2AK2 P19525 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6506758 0.76 IKBKB (0.50) MAPTIKBKBJAK2JAK3CHEK1
SCHEMBL6514861 0.73 DYRK1A (0.52) MAPTIKBKBJAK2JAK3
SCHEMBL27570742 0.72 HTR3E (0.69) HSD17B1HSD17B2HTR3EHTR3BHTR3A
SCHEMBL6507152 0.71 IKBKB (0.57) TDP1IKBKBJAK2JAK3CHEK1
SCHEMBL6506340 0.69 FLT3 (0.51) TDP1MAPTIKBKBJAK2JAK3
SCHEMBL6505865 0.68 IKBKB (0.58) TDP1IKBKBJAK2JAK3CHEK1
SCHEMBL7368760 0.68 HTR3E (0.54) HSD17B1HSD17B2HTR3EHTR3BHTR3A
SCHEMBL6629827 0.68 HTR3E (0.61) HSD17B1HSD17B2HTR3EHTR3BHTR3A
SCHEMBL6505484 0.68 CHEK1 (0.55) TDP1IKBKBJAK2JAK3CHEK1
SCHEMBL6510565 0.68 MAPK8 (0.65) TDP1IKBKBJAK2JAK3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed