SCHEMBL7368760

SCHEMBL7368760

CN(C(=O)c1ccc(N)cc1)c1cccc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.54
HTR3B O95264 1/20 0.54
HTR3A P46098 1/20 0.54
HTR3D Q70Z44 1/20 0.54
HTR3C Q8WXA8 1/20 0.54
HSD17B1 P14061 7/20 0.50
HSD17B2 P37059 7/20 0.50
TP53 P04637 1/20 0.48
KMT2A Q03164 2/20 0.46
MAPT P10636 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
GPBAR1 Q8TDU6 1/20 0.44
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAOA P21397 1/20 0.43
PLAU P00749 1/20 0.43
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18585572 0.86 ATF1 (0.42) HSD17B1HSD17B2KMT2AEGFRERBB2
SCHEMBL7374140 0.83 HSD17B1 (0.71) HSD17B1HSD17B2HTTKDM4ENPC1
SCHEMBL7410067 0.81 CHEK2 (0.49) TP53KMT2AMAPTTDP1GPBAR1
SCHEMBL7373511 0.80 KMT2A (0.64) KMT2AEGFRERBB2HTTKDM4E
SCHEMBL7368659 0.80 ATM (0.57) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7376609 0.79 HSD17B2 (0.75) HSD17B1HSD17B2
SCHEMBL18585586 0.79 GPBAR1 (0.39) HSD17B1HSD17B2KMT2AGPBAR1EGFR
SCHEMBL8581201 0.78 KMT2A (0.50) HSD17B1HSD17B2TP53KMT2AMAPT
SCHEMBL2127770 0.78 KMT2A (0.50) HSD17B1HSD17B2TP53KMT2AMAPT
SCHEMBL4250786 0.78 HTR3E (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed