SCHEMBL6511078

SCHEMBL6511078

CCC(C)c1ccc(N=C(N)Nc2cc(C)cc(C)n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 3/20 0.43
GRIN3B O60391 3/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2A Q12879 3/20 0.43
GRIN2B Q13224 3/20 0.43
GRIN2C Q14957 3/20 0.43
GRIN3A Q8TCU5 3/20 0.43
SIGMAR1 Q99720 3/20 0.43
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2C9 P11712 1/20 0.39
LMNA P02545 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
CRHBP P24387 2/20 0.38
CRHR2 Q13324 2/20 0.38
CYP1A2 P05177 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4979589 0.76 SIGMAR1 (0.71) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL5923056 0.76 SMN1; SMN2 (0.45) MAPK1ALDH1A1SMN1; SMN2LMNACHRNB2
SCHEMBL6518566 0.74 CYP1A2 (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6515597 0.73 NOS3 (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6515320 0.71 SIGMAR1 (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6510602 0.67 MAPK1 (0.63) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6513329 0.67 MAPK1 (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL15938854 0.65 RAC1 (0.67) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6507381 0.64 RAB9A (0.54) MAPK1SMN1; SMN2LMNACHRNB2CHRNB4
SCHEMBL6508707 0.64 KMT2A (0.60) MAPK1ALDH1A1SMN1; SMN2LMNACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed