SCHEMBL6515320

SCHEMBL6515320

Cc1cc(C)nc(NC(N)=Nc2cccc(Cc3ccccc3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.46
GRIN2D O15399 3/20 0.46
GRIN3B O60391 3/20 0.46
GRIN1 Q05586 3/20 0.46
GRIN2A Q12879 3/20 0.46
GRIN2B Q13224 3/20 0.46
GRIN2C Q14957 3/20 0.46
GRIN3A Q8TCU5 3/20 0.46
PHGDH O43175 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 2/20 0.42
NOS1 P29475 1/20 0.41
POLB P06746 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CRHBP P24387 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510588 0.84 LMNA (0.50) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6510602 0.84 MAPK1 (0.63) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6507964 0.78 SIGMAR1 (0.72) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6507347 0.75 LMNA (0.52) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6508617 0.74 SIGMAR1 (0.46) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6507406 0.74 RAB9A (0.52) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5923236 0.74 SMN1; SMN2 (0.50) PHGDHSMN1; SMN2ALDH1A1MAPK1RAB9A
SCHEMBL6510249 0.72 MAPK1 (0.62) SIGMAR1SMN1; SMN2ALDH1A1MAPK1POLB
SCHEMBL6513739 0.72 SMN1; SMN2 (0.42) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL14861786 0.72 SIGMAR1 (0.65) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed