SCHEMBL6511368

SCHEMBL6511368

CC1(C)CC(=C(c2ccc(O)cc2)c2c(C(N)=O)cccc2-c2ccccc2)CC(C)(C)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.42
MMP9 P14780 1/20 0.38
ESR1 P03372 1/20 0.38
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
PLAU P00749 1/20 0.35
PLAT P00750 1/20 0.35
HNF4A P41235 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PARP1 P09874 2/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
MYC P01106 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27640751 0.82 ESR1 (0.39) BCAT2MMP9ESR1HNF4ASCN1A
SCHEMBL3467813 0.81 ESR1 (0.44) MMP9ESR1HNF4ARAB9AMYC
SCHEMBL3468563 0.76 MMP3 (0.47) ESR1NPC1RAB9AMEN1KMT2A
SCHEMBL3468554 0.76 ESR1 (0.54) ESR1PARP1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL3468373 0.76 SLC6A3 (0.49) ESR1SCN1ASCN2ASCN3AALDH1A1
SCHEMBL3468462 0.75 ESR1 (0.43) ESR1PLAUPLATPARP1MEN1
SCHEMBL3075044 0.74 ESR1 (0.50) ESR1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL3468030 0.73 ESR1 (0.40) MMP9ESR1PDCD1CD274NPC1
Gsk-232802 SCHEMBL3467757 0.71 ESR1 (0.55) ESR1HNF4AMEN1KMT2ASMN1; SMN2
SCHEMBL3468706 0.71 KMO (0.47) ESR1RAB9AMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005012220-A9 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF ESTROGEN RECEPTOR SMITHKLINE BEECHAM CORP (US) 2005-05-19 WO disclosed