SCHEMBL6522029

SCHEMBL6522029

C[C](C)Cc1ccc(O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.54
CAMK2A Q9UQM7 1/20 0.54
ESR1 P03372 4/20 0.52
ESR2 Q92731 2/20 0.52
ALDH1A1 P00352 2/20 0.48
FNTA P49354 1/20 0.48
FNTB P49356 1/20 0.48
PKM P14618 1/20 0.48
ABAT P80404 1/20 0.48
TAAR1 Q96RJ0 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
CA12 O43570 1/20 0.44
GMNN O75496 1/20 0.44
CA1 P00915 1/20 0.44
LMNA P02545 1/20 0.44
CA3 P07451 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10702370 0.81 CA2 (0.58) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL465583 0.79 CA2 (0.50) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL10629788 0.79 CA2 (0.60) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL4455 0.79 CA2 (0.62) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL6616424 0.78 LPL (0.48) CA2ALDH1A1TAAR1
SCHEMBL4226247 0.78 IDO1 (0.48) ALDH1A1TAAR1MEN1NPC1LMNA
SCHEMBL2459593 0.77 CA2 (0.48) CA2CAMK2AESR1ESR2ALDH1A1
Hydrochloric Acid SCHEMBL2583907 0.77 CA2 (0.60) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL9261880 0.77 CA2 (0.48) CA2CAMK2AESR1ESR2ALDH1A1
SCHEMBL1620786 0.76 TDP1 (0.47) ALDH1A1TAAR1KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050112693-A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof NEFZI ADEL (US) 2005-05-26 US claimed
US-20030120066-A1 Synthetic peptides NEFZI ADEL (US) 2003-06-26 US claimed
US-5364948-A Anticancer, anticholesterol, fungicide MERCK & CO., INC. (US) 1994-11-15 US claimed
EP-0002792-A1 3-Aminopropoxyaryl derivatives, their preparation and pharmaceutical compositions containing them SANDOZ AG (CH) 1979-07-11 EP claimed
CN-1713914-A Novel drug for treating chronic obstructive pulmonary disease BOEHRINGER INGELHEIM PHARMA (DE) 2005-12-28 CN disclosed
US-6809202-B2 SYNTHETIC PEPTIDES TORREY PINES INSTITUTE FOR MOLECULAR STUDIES 2004-10-26 US disclosed
WO-2004046080-A1 METHOD OF PREPARATION OF DERIVATIVES OF SUBSTITUTED 2-ARYL AIKANOIC ACIDS ZENTIVA, A.S. (SK) 2004-06-03 WO disclosed
US-20030120066-A1 Synthetic peptides NEFZI ADEL (US) 2003-06-26 US disclosed
US-5811422-A USEFUL FOR TREATING VIRAL INFECTIONS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-09-22 US disclosed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US disclosed
US-5434164-A Carbostyril derivatives and salts thereof and pharmaceutical compositions for inhibiting adhesion of thrombocytes OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1995-07-18 US disclosed
EP-0240015-B1 Carbostyril derivatives, process for preparing them, pharmaceutical composition, and use OTSUKA PHARMA CO LTD (JP) 1994-12-28 EP disclosed
US-4148908-A BRONCHODILATORS MEAD JOHNSON & COMPANY (US) 1979-04-10 US disclosed
US-4119729-A TREATMENT OF HYPERTENSION MEAD JOHNSON & COMPANY (US) 1978-10-10 US disclosed
US-4104402-A BRONCHODILATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1978-08-01 US disclosed
US-4067904-A ANTIARRHYTHMIA, HYPOTENSIVE MEAD JOHNSON & COMPANY (US) 1978-01-10 US disclosed
US-4055658-A BETA-ADRENERGIC STIMULANTS, BRONCHIAL MEAD JOHNSON & COMPANY (US) 1977-10-25 US disclosed
US-4048229-A ANTAGONIST ACTIVITY SMITHKLINE CORPORATION (US) 1977-09-13 US disclosed
US-4035512-A Aminotetralols TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-07-12 US disclosed
US-4010202-A TREATMENT OF ASTHMA AND ARRHYTHMIA TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050112693-A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof DHPS, DCK, DAZAP1 CA2 2644/4885CAMK2A 2606/4885ESR1 4384/4885
US-20030120066-A1 Synthetic peptides VIP, NGLY1, GRPR CA2 3987/4885CAMK2A 4375/4885ESR1 4195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.