SCHEMBL6522590

SCHEMBL6522590

CN1CCc2ccccc2C1.O=S(=O)(O)c1ccccc1

nearest known ligand 0.67

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 1/20 0.52
MAOA P21397 2/20 0.67
MAOB P27338 2/20 0.67
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
TSHR P16473 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
DRD1 P21728 2/20 0.52
DRD5 P21918 2/20 0.52
DRD4 P21917 1/20 0.52
DRD3 P35462 1/20 0.52
HTR7 P34969 6/20 0.50
LMNA P02545 2/20 0.50
HPGD P15428 1/20 0.50
THRB P10828 1/20 0.49
PMP22 Q01453 1/20 0.49
HSD17B10 Q99714 1/20 0.49
POLB P06746 1/20 0.49
AKR1C3 P42330 2/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL6520165 0.90 MAOA (0.77) MAOAMAOBMEN1KMT2ATSHR
SCHEMBL6524885 0.89 MAOA (0.61) MAOAMAOBMEN1KMT2ATSHR
Sulfuric Acid SCHEMBL6520169 0.85 MAOA (0.69) MAOAMAOBMEN1KMT2ATSHR
Sulfuric Acid SCHEMBL174314 0.84 DRD1 (0.65) MAOAMAOBTSHRDRD1DRD5
SCHEMBL22283827 0.83 TSHR (0.57) MAOAMAOBTSHRSMN1; SMN2DRD1
SCHEMBL29390912 0.82 MAOA (1.00) MAOAMAOBDRD1DRD5DRD2
SCHEMBL98108 0.82 MAOA (1.00) MAOAMAOBDRD1DRD5DRD2
N-Methyl Pyrrolidine (Nmp) SCHEMBL1374351 0.80 TSHR (0.64) TSHRSMN1; SMN2LMNAHPGDPOLB
SCHEMBL6521382 0.80 HTR7 (0.61) MEN1KMT2ADRD2DRD3HTR7
Hydrochloric Acid SCHEMBL23501375 0.80 MAOA (1.00) MAOAMAOBDRD1DRD5DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274056-B1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOCHINOLINIUM DERIVATIVES, SPECIFIC ALKANOLAMINES AND HYDROGEN PEROXYDE HENKEL AG & CO KGAA (DE) 2012-10-03 EP claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE KRT18, H1-3, H1-2 DRD2 791/4885MAOA 74/4885MAOB 66/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.