SCHEMBL6522652

SCHEMBL6522652

N#Cc1ccc(C(Cc2ccc(C(F)(F)F)cn2)Cc2nc[nH]n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.42
KIF11 P52732 1/20 0.36
MAOB P27338 2/20 0.36
VNN1 O95497 2/20 0.35
DAO P14920 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
KDM1A O60341 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP3A5 P20815 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
CNR1 P21554 2/20 0.32
KMT2A Q03164 1/20 0.32
CCR6 P51684 1/20 0.32
DGAT1 O75907 1/20 0.31
SOAT1 P35610 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6474489 0.85 CYP19A1 (0.44) CYP19A1KIF11MAOBVNN1DAO
SCHEMBL6526163 0.77 CYP19A1 (0.41) CYP19A1MAOBALDH1A1
SCHEMBL6527102 0.75 TRPA1 (0.40) CYP19A1MAOBPTGDR2KDM1AALDH1A1
SCHEMBL2350966 0.74 CYP19A1 (0.43) CYP19A1KIF11MAOBCYP3A4CYP3A5
SCHEMBL9159563 0.70 KIF11 (0.47) CYP19A1KIF11MAOBVNN1PTGDR2
SCHEMBL9192710 0.66 CYP19A1 (0.45) CYP19A1VNN1PTGDR2
SCHEMBL6573450 0.65 CYP19A1 (0.41) CYP19A1MAOBVNN1PTGDR2
SCHEMBL11092221 0.64 GABBR2 (0.34) CYP19A1CYP3A4KMT2A
SCHEMBL9093244 0.64 CYP19A1 (0.61) CYP19A1KIF11MAOBVNN1PTGDR2
SCHEMBL5925435 0.64 KIF11 (0.43) CYP19A1KIF11MAOBVNN1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534265-A1 COMBINATION OF AN AROMATASE INHIBITOR WITH A BISPHOSPHONATE Novartis AG (CH) 2005-06-01 EP disclosed
WO-2004012728-A1 COMBINATION OF AN AROMATASE INHIBITOR WITH A BISPHOSPHONATE NOVARTIS AG (CH) 2004-02-12 WO disclosed