SCHEMBL6527434

SCHEMBL6527434

O=C1c2ccccc2C(=O)N1Cc1cn(-c2cc(F)c(C3=CCNCC3)c(F)c2)nn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 5/20 0.39
HTR6 P50406 4/20 0.39
ACHE P22303 1/20 0.38
MAPT P10636 1/20 0.35
RECQL P46063 1/20 0.35
PTGS2 P35354 2/20 0.35
ALOX15 P16050 1/20 0.35
DRD3 P35462 2/20 0.35
AMY1A P0DUB6 2/20 0.35
HTR1A P08908 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
PARP1 P09874 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528580 0.90 HTR6 (0.40) TYRHTR6ACHEPTGS2ALOX15
SCHEMBL6920471 0.83 TYR (0.39) TYRACHEMAPTRECQLPTGS2
SCHEMBL6529962 0.76 GRM5 (0.39) TYRACHEDRD3DRD2DRD4
SCHEMBL6529525 0.75 GRM1 (0.55) HTR6
SCHEMBL6925271 0.72 TYR (0.38) TYRACHEMAPTRECQLPTGS2
SCHEMBL6533328 0.72 MAPT (0.41) TYRMAPTDRD3AMY1AHTR1A
SCHEMBL6528269 0.69 GRM1 (0.41) TYRPTGS2ALOX15DRD3HTR1A
SCHEMBL5623713 0.69 ALDH1A1 (0.45) TYRMAPTALOX15ALDH1A1
SCHEMBL6532725 0.68 TYR (0.39) TYRACHEPTGS2ALOX15DRD3
SCHEMBL6527437 0.67 CDK9 (0.34) HTR6MAPTALOX15DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed