SCHEMBL6528929

SCHEMBL6528929

CCOc1ccc2c(c1)c(C1=C(Cl)CN(C)C1)cn2S(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.56
CYP2D6 P10635 4/20 0.56
HTR6 P50406 17/20 0.50
HTR2A P28223 2/20 0.41
DRD2 P14416 1/20 0.40
HTR7 P34969 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
KLK7 P49862 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528108 0.89 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6530751 0.83 CYP3A4 (0.64) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6529028 0.79 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6529121 0.79 CYP3A4 (0.74) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6527747 0.78 HTR6 (0.62) CYP3A4CYP2D6HTR6HTR2A
SCHEMBL6528427 0.78 CYP3A4 (0.57) CYP3A4CYP2D6HTR6HTR2A
SCHEMBL6532617 0.76 CYP3A4 (0.79) CYP3A4CYP2D6HTR6
SCHEMBL6529764 0.74 HTR6 (0.61) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL5667148 0.73 PPARG (0.71) HTR6DRD2HTR7
SCHEMBL6527092 0.72 CYP3A4 (1.00) CYP3A4CYP2D6HTR6HTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005066157-A1 3-(PYROLIDIN-3-L) INDOLES AS 5-HT6 RECEPTOR MODULATORS SUVEN LIFE SCIENCES (IN) 2005-07-21 WO claimed
WO-2005066157-A1 3-(PYROLIDIN-3-L) INDOLES AS 5-HT6 RECEPTOR MODULATORS SUVEN LIFE SCIENCES (IN) 2005-07-21 WO disclosed