SCHEMBL6530751

SCHEMBL6530751

COc1ccc(S(=O)(=O)n2cc(C3=C(Cl)CN(C)C3)c3cc(OC)ccc32)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.64
CYP2D6 P10635 6/20 0.64
HTR6 P50406 17/20 0.57
HTR2A P28223 2/20 0.52
PPARG P37231 2/20 0.51
PPARD Q03181 2/20 0.51
PPARA Q07869 2/20 0.51
HTR1A P08908 1/20 0.50
DRD2 P14416 1/20 0.48
HTR7 P34969 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529028 0.94 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2AHTR1A
SCHEMBL6528108 0.94 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2APPARG
SCHEMBL6529121 0.94 CYP3A4 (0.74) CYP3A4CYP2D6HTR6HTR2AHTR1A
SCHEMBL6527747 0.93 HTR6 (0.62) CYP3A4CYP2D6HTR6HTR2AHTR1A
SCHEMBL6532617 0.90 CYP3A4 (0.79) CYP3A4CYP2D6HTR6
SCHEMBL6530026 0.86 CYP3A4 (0.52) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6528427 0.83 CYP3A4 (0.57) CYP3A4CYP2D6HTR6HTR2A
SCHEMBL6529764 0.83 HTR6 (0.61) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6528929 0.83 CYP3A4 (0.56) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6533974 0.81 HTR6 (0.62) CYP3A4CYP2D6HTR6HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005066157-A1 3-(PYROLIDIN-3-L) INDOLES AS 5-HT6 RECEPTOR MODULATORS SUVEN LIFE SCIENCES (IN) 2005-07-21 WO disclosed