SCHEMBL6529121

SCHEMBL6529121

COc1ccc2c(c1)c(C1=C(Cl)CN(C)C1)cn2S(=O)(=O)c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.74
CYP2D6 P10635 1/20 0.74
HTR6 P50406 19/20 0.58
HTR2A P28223 4/20 0.56
DRD2 P14416 4/20 0.56
HTR7 P34969 3/20 0.56
HTR1A P08908 1/20 0.53
HTR1D P28221 1/20 0.53
HTR1B P28222 1/20 0.53
HTR1E P28566 1/20 0.53
HTR1F P30939 1/20 0.53
DRD3 P35462 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530751 0.94 CYP3A4 (0.64) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6529028 0.90 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6528108 0.90 HTR6 (0.60) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6527747 0.89 HTR6 (0.62) CYP3A4CYP2D6HTR6HTR2AHTR1A
SCHEMBL6532617 0.88 CYP3A4 (0.79) CYP3A4CYP2D6HTR6
SCHEMBL6533974 0.88 HTR6 (0.62) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6529764 0.86 HTR6 (0.61) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6527092 0.85 CYP3A4 (1.00) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL6530026 0.84 CYP3A4 (0.52) CYP3A4CYP2D6HTR6HTR2ADRD2
SCHEMBL19737472 0.81 HTR6 (0.66) HTR6HTR2ADRD2HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005066157-A1 3-(PYROLIDIN-3-L) INDOLES AS 5-HT6 RECEPTOR MODULATORS SUVEN LIFE SCIENCES (IN) 2005-07-21 WO disclosed