SCHEMBL6532745

SCHEMBL6532745

NC(=O)Nc1cnc(Cl)c(-c2cccs2)c1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.41
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
KDM4E B2RXH2 7/20 0.40
ALDH1A1 P00352 6/20 0.40
GAA P10253 5/20 0.40
HSD17B10 Q99714 4/20 0.40
MAPT P10636 4/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 2/20 0.40
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
RAB9A P51151 4/20 0.38
POLB P06746 1/20 0.37
NPC1 O15118 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
CHEK1 O14757 1/20 0.36
CHEK2 O96017 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4314650 0.70 KDM4E (0.43) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL6532748 0.70 ADORA2A (0.42) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL4341035 0.67 KDM4E (0.44) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL1385872 0.65 IKBKB (0.67) KDM4EMAPTKMT2ANPC1NPSR1
SCHEMBL6532742 0.64 NR3C1 (0.44) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL5554748 0.62 IKBKB (0.58) KDM4EMAPTKMT2AMEN1POLB
SCHEMBL30174203 0.62 ERCC1 (0.46) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL6533212 0.62 PARP1 (0.44) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL4092063 0.62 KIF11 (0.51) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL15109937 0.62 KDM4E (0.44) KDM4EALDH1A1GAAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed