SCHEMBL6535680

SCHEMBL6535680

Pc1cccc2c1-c1ccccc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
MAPK1 P28482 3/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ATM Q13315 1/20 0.39
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
MAPT P10636 3/20 0.36
PTPRC P08575 3/20 0.36
LMNA P02545 2/20 0.36
S100A4 P26447 2/20 0.36
KDM4E B2RXH2 2/20 0.36
CES2 O00748 1/20 0.36
APAF1 O14727 1/20 0.36
TERT O14746 1/20 0.36
NPC1 O15118 1/20 0.36
PLIN1 O60240 1/20 0.36
TDP2 O95551 1/20 0.36
S1PR4 O95977 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9927308 0.84 MAOA (0.32) ALDH1A1MAPK1L3MBTL1TSHRHSD17B10
SCHEMBL29236876 0.81 ALDH1A1 (0.47) ALDH1A1MAPK1L3MBTL1TSHRHSD17B10
SCHEMBL476858 0.78 APP (0.57) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7323816 0.78 TSHR (0.39) ALDH1A1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL5596876 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1L3MBTL1TSHRHSD17B10
SCHEMBL9324952 0.78 ALDH1A1 (0.59) ALDH1A1L3MBTL1TSHRHSD17B10MEN1
SCHEMBL2454271 0.78 CYP2A6 (0.44) ALDH1A1TSHRKMT2APTPRCLMNA
SCHEMBL22831361 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1L3MBTL1TSHRHSD17B10
SCHEMBL4061121 0.78 HNF4A (0.39) ALDH1A1MAPK1HSD17B10MAPTLMNA
SCHEMBL1752721 0.74 MEN1 (0.39) ALDH1A1MAPK1L3MBTL1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6437164-B1 REACTING BIPHENYL AND PHOSPHORUS TRICHLORIDE IN PRESENCE OF ALUMINUM CHLORIDE, ADDING PYRIDINE, RESULTING DICHLOROPHOSPHINE IS REACTED WITH A PHENOL, REMOVING FORMED PYRIDINE-ALUMINUM CHLORIDE COMPLEX YOSHITOMI FINE CHEMICALS, LTD. (JP) 2002-08-20 US claimed
EP-1142898-A1 PROCESS FOR THE PREPARATION OF PHOSPHONITE COMPOUNDS Yoshitomi Fine Chemicals, Ltd. (JP) 2001-10-10 EP claimed
EP-0114904-B1 STABILIZED CARBOXYL-CONTAINING ETHYLENE INTERPOLYMERS THE DOW CHEMICAL COMPANY (US) 1987-11-19 EP claimed
EP-0114904-A1 Stabilized carboxyl-containing ethylene interpolymers THE DOW CHEMICAL COMPANY (US) 1984-08-08 EP claimed
CN-102812072-B Film 帝人株式会社 2016-10-19 CN disclosed
CN-1898253-A Method for producing trivalent organophosphorus compounds OXENO OLEFINCHEMIE GMBH (DE) 2007-01-17 CN disclosed
EP-1142898-A4 PROCESS FOR THE PREPARATION OF PHOSPHONITE COMPOUNDS API CORP (JP) 2004-09-01 EP disclosed
US-6437164-B1 REACTING BIPHENYL AND PHOSPHORUS TRICHLORIDE IN PRESENCE OF ALUMINUM CHLORIDE, ADDING PYRIDINE, RESULTING DICHLOROPHOSPHINE IS REACTED WITH A PHENOL, REMOVING FORMED PYRIDINE-ALUMINUM CHLORIDE COMPLEX YOSHITOMI FINE CHEMICALS, LTD. (JP) 2002-08-20 US disclosed
US-6437164-B1 REACTING BIPHENYL AND PHOSPHORUS TRICHLORIDE IN PRESENCE OF ALUMINUM CHLORIDE, ADDING PYRIDINE, RESULTING DICHLOROPHOSPHINE IS REACTED WITH A PHENOL, REMOVING FORMED PYRIDINE-ALUMINUM CHLORIDE COMPLEX YOSHITOMI FINE CHEMICALS, LTD. (JP) 2002-08-20 US disclosed
EP-1142898-A1 PROCESS FOR THE PREPARATION OF PHOSPHONITE COMPOUNDS Yoshitomi Fine Chemicals, Ltd. (JP) 2001-10-10 EP disclosed
EP-1142898-A1 PROCESS FOR THE PREPARATION OF PHOSPHONITE COMPOUNDS Yoshitomi Fine Chemicals, Ltd. (JP) 2001-10-10 EP disclosed
CN-1056860-C Copolymeric polyamide and preparation of same TORAY INDUSTRIES (JP) 2000-09-27 CN disclosed
WO-2000040587-A1 PROCESS FOR THE PREPARATION OF PHOSPHONITE COMPOUNDS YOSHITOMI FINE CHEMICALS, LTD. (JP) 2000-07-13 WO disclosed
CN-1127266-A Copolymeric polyamide and preparation of same TORAY INDUSTRIES (JP) 1996-07-24 CN disclosed
EP-0114904-B1 STABILIZED CARBOXYL-CONTAINING ETHYLENE INTERPOLYMERS THE DOW CHEMICAL COMPANY (US) 1987-11-19 EP disclosed
EP-0114904-A1 Stabilized carboxyl-containing ethylene interpolymers THE DOW CHEMICAL COMPANY (US) 1984-08-08 EP disclosed
EP-0114904-A1 Stabilized carboxyl-containing ethylene interpolymers THE DOW CHEMICAL COMPANY (US) 1984-08-08 EP disclosed