SCHEMBL6535836

SCHEMBL6535836

O=C(O)c1[nH]c2cccc(Cc3ccc(Cl)cc3)c2c1C1=CC(=S)CC(Cl)=C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 5/20 0.37
MAP2 P11137 1/20 0.36
GPR35 Q9HC97 2/20 0.35
HRH1 P35367 1/20 0.34
MDM4 O15151 2/20 0.33
MDM2 Q00987 2/20 0.33
TP53 P04637 1/20 0.33
GRIN1 Q05586 1/20 0.33
FBP1 P09467 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
MCL1 Q07820 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9457645 0.75 KDM4E (0.57) MAP2GPR35KDM4EALDH1A1HPGD
SCHEMBL7694143 0.64 MAPT (0.49) TP53KDM4EALDH1A1
SCHEMBL7074273 0.62 MDM2 (0.40) GPR17MDM2MCL1
SCHEMBL8647087 0.62 NPSR1 (0.40) HRH1KDM4EALDH1A1
SCHEMBL7698766 0.62 ALDH1A1 (0.38) HRH1KDM4EALDH1A1
SCHEMBL8543287 0.61 MAP2 (0.42) MAP2KDM4EALDH1A1HPGD
SCHEMBL5778905 0.61 GPR35 (0.49) GPR17MAP2GPR35KDM4EALDH1A1
SCHEMBL9816507 0.60 KDM4E (0.79) MAP2GPR35MDM4MDM2KDM4E
SCHEMBL7463695 0.60 SLC6A2 (0.41) GPR17GRIN1MCL1
SCHEMBL5214867 0.59 ALOX5 (0.47) TP53ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284728-A4 PHARMACEUTICALS FOR TREATING OBESITY MERCK & CO INC (US) 2004-05-19 EP disclosed
EP-1284728-A1 PHARMACEUTICALS FOR TREATING OBESITY Merck & Co., Inc. (US) 2003-02-26 EP disclosed
WO-2001030343-A1 PHARMACEUTICALS FOR TREATING OBESITY MERCK & CO., INC. (US) 2001-05-03 WO disclosed