SCHEMBL6542003

SCHEMBL6542003

Cc1cc2c(cc1-c1ccc(C=O)cn1)C(C)(C)CCC2(C)C

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RXRA P19793 16/20 0.44
RARG P13631 8/20 0.44
RXRG P48443 10/20 0.43
RXRB P28702 9/20 0.43
RARB P10826 7/20 0.41
RARA P10276 7/20 0.40
PPARG P37231 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6542008 0.83 RXRA (0.42) RXRARARGRXRGRXRBRARB
SCHEMBL26240347 0.81 CCR1 (0.46) RXRARARGRXRGRXRBRARB
SCHEMBL6542688 0.79 RXRA (0.52) RXRARARGRXRGRXRBRARB
SCHEMBL13480474 0.76 RXRA (0.65) RXRARARGRXRGRXRBRARB
SCHEMBL6032609 0.75 RXRA (0.38) RXRARARGRXRGRXRBRARB
SCHEMBL5483831 0.75 RXRA (0.42) RXRARARGRXRGRXRBRARB
SCHEMBL21976175 0.75 RARG (0.44) RXRARARGRXRGRXRBRARB
SCHEMBL6543042 0.75 RXRA (0.58) RXRARARGRXRGRXRBRARB
SCHEMBL6541444 0.74 ALDH1A1 (0.47) RXRARARGRXRGRXRBRARB
SCHEMBL5486511 0.74 RXRA (0.71) RXRARARGRXRGRXRBRARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421061-A4 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA INCYTE SAN DIEGO INC (US) 2004-12-22 EP disclosed
EP-1421061-A1 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA Incyte San Diego Incorporated (US) 2004-05-26 EP disclosed
US-20030083357-A1 Oxime derivatives for the treatment of dyslipidemia and hypercholesteremia ORTHO MCNEIL PHARMACEUTICAL INC. 2003-05-01 US disclosed
WO-2003016267-A1 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA INCYTE SAN DIEGO INCORPORATED (US) 2003-02-27 WO disclosed
EP-1214305-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION Maxia Pharmaceuticals, Inc. (US) 2002-06-19 EP disclosed
WO-2001016123-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION MAXIA PHARMACEUTICALS, INC. (US) 2001-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030083357-A1 Oxime derivatives for the treatment of dyslipidemia and hypercholesteremia OAT, CPT1A, CYP27A1 RXRA 793/4885RARG 1440/4885RXRG 744/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.