SCHEMBL6545705

SCHEMBL6545705

Cc1ccc(S(=O)(=O)OC(=O)[C@@H](N)CCCCNC(=O)[C@@H](N)Cc2cn(S(=O)(=O)c3ccc(C)cc3)c3ccccc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDE P14735 1/20 0.55
HTR6 P50406 8/20 0.47
ALK Q9UM73 1/20 0.43
ALOX5 P09917 7/20 0.43
PTGS2 P35354 2/20 0.42
DRD2 P14416 1/20 0.41
CYP19A1 P11511 1/20 0.41
KDM4E B2RXH2 1/20 0.39
UBE2N P61088 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL838017 0.77 HTR6 (0.64) IDEHTR6ALKALOX5PTGS2
SCHEMBL838015 0.77 HTR6 (0.64) IDEHTR6ALKALOX5PTGS2
SCHEMBL7583708 0.72 HTR6 (0.51) IDEHTR6ALKALOX5PTGS2
SCHEMBL10365920 0.72 DPP8 (0.55)
SCHEMBL28381352 0.70 ITGB3 (0.42) KDM4E
SCHEMBL27498945 0.70 ITGB3 (0.42) KDM4E
SCHEMBL7588756 0.70 IDE (0.47) IDEHTR6ALKALOX5PTGS2
SCHEMBL29169604 0.70 HTR6 (0.69) HTR6ALKDRD2CYP19A1KDM4E
SCHEMBL14286783 0.69 ALOX5 (0.55) HTR6ALKALOX5PTGS2CYP19A1
SCHEMBL29169606 0.69 HTR6 (0.67) IDEHTR6ALKALOX5PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377542-A1 HIV PROTEASE INHIBITORS BASED ON AMINO ACID DERIVATIVES Pharmacor Inc. (CA) 2004-01-07 EP disclosed
WO-2002064551-A1 HIV PROTEASE INHIBITORS BASED ON AMINO ACID DERIVATIVES PHARMACOR INC. (CA) 2002-08-22 WO disclosed