SCHEMBL6547586

SCHEMBL6547586

COc1cccc(N=C(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.62
HTR3B O95264 1/20 0.62
HTR3A P46098 1/20 0.62
HTR3D Q70Z44 1/20 0.62
HTR3C Q8WXA8 1/20 0.62
TAAR1 Q96RJ0 1/20 0.60
SIGMAR1 Q99720 1/20 0.53
NOS3 P29474 2/20 0.51
NOS1 P29475 2/20 0.51
NOS2 P35228 2/20 0.51
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
NLRP3 Q96P20 1/20 0.50
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
MITF O75030 1/20 0.47
LMNA P02545 1/20 0.47
AGTR1 P30556 1/20 0.47
OPRK1 P41145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608124 0.86 NPC1 (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11378646 0.83 HTR3E (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11378649 0.83 HTR3E (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL11776533 0.82 TAAR1 (0.69) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9370892 0.81 HTR3E (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9370900 0.81 HTR3E (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6548684 0.80 NOS3 (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL19505630 0.80 ESR1 (0.60) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL12077531 0.77 MEN1 (0.59) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL2944424 0.77 HTR3E (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100774-B1 IMPROVED ARYLAMINE SYNTHESIS MASSACHUSETTS INST TECHNOLOGY (US) 2004-01-21 EP disclosed
US-6323366-B1 ACTIVATED ARYL GROUP AND AN IMINE GROUP ARE COMBINED, IN THE PRESENCE OF A TRANSITION METAL CATALYST FOR FORMATION OF A CARBON-NITROGEN BOND BETWEEN THE ACTIVATED CARBON OF THE ARENE AND IMINE NITROGEN; CONVERTING TO ARYLAMINE MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-11-27 US disclosed