SCHEMBL6551932

SCHEMBL6551932

COc1nn(-c2ccc(S(=O)(=O)NC(C)N(C(C)C)C(C)C)cc2)c(=O)o1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABHD16A O95870 2/20 0.53
FAAH O00519 13/20 0.49
MGLL Q99685 7/20 0.49
LPL P06858 1/20 0.43
LIPC P11150 1/20 0.43
LIPE Q05469 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6551212 0.91 ABHD16A (0.41) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL7040759 0.74 ABHD16A (0.58) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL2233598 0.73 ABHD16A (0.72) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL6599976 0.71 LMNA (0.56) ABHD16AFAAHMGLL
SCHEMBL6551927 0.71 KMT2A (0.52) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL2233406 0.70 ABHD16A (0.72) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL7046228 0.70 ABHD16A (0.72) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL11620781 0.70 FAAH (0.78) ABHD16AFAAHMGLLLPLLIPC
SCHEMBL6552647 0.70 ABHD16A (0.55) ABHD16AFAAHMGLL
SCHEMBL6551881 0.70 ABHD16A (0.55) ABHD16AFAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1482929-A1 USE OF SUBSTITUTED 3-PHENYL-5-ALKOXY-1,3,4-OXDIAZOLE-2-ONE FOR PRODUCING MEDICAMENTS THAT INHIBIT PANCREATIC LIPASE Aventis Pharma Deutschland GmbH (DE) 2004-12-08 EP disclosed
EP-1214302-B1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS AVENTIS PHARMA GMBH (DE) 2003-10-29 EP disclosed
WO-2003072098-A1 USE OF SUBSTITUTED 3-PHENYL-5-ALKOXY-1,3,4-OXDIAZOLE-2-ONE FOR PRODUCING MEDICAMENTS THAT INHIBIT PANCREATIC LIPASE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-09-04 WO disclosed
US-6596742-B1 Inhibitory effect on the hormone-sensitive lipase, HSL. insecticides, controlling metabolism and multistage synthesis AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-07-22 US disclosed
EP-1214302-A1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS Aventis Pharma Deutschland GmbH (DE) 2002-06-19 EP disclosed
WO-2001017981-A1 SUBSTITUTED 3-PHENYL-5-ALKOXI-1,3,4-OXDIAZOL-2-ONES AND THEIR USE AS LIPASE INHIBITORS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-15 WO disclosed